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(±)-BI-D
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(±)-BI-D

$525.00$3,150.00

(±)-BI-D is a potent ALLINI (An allosteric IN inhibitor) that binds integrase at the LEDGF/p75 binding site.

(R)-(+)-Etomoxir (sodium salt)
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(R)-(+)-Etomoxir (sodium salt)

$141.00$738.50

(R)- (+)-Etomoxir (sodium salt) is a potent inhibitor of carnitine palmitoyltransferase I (CPT1); inhibits ?-oxidation in mitochondria; shown to inhibit cardiolipin biosynthesis from exogenous fatty acid in H9c2 cells.

17-AAG
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17-AAG

$99.00$505.00

17-AAG (NSC 330507; CP 127374) is a potent HSP90 inhibitor with IC50 of 5 nM, having a 100-fold higher binding affinity for HSP90 derived from tumour cells than HSP90 from normal cells.

17-AAG (Hydrochloride)
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17-AAG (Hydrochloride)

$99.00$505.00

17-AAG Hcl is a potent HSP90 inhibitor with IC50 of 5 nM, having a 100-fold higher binding affinity for HSP90 derived from tumour cells than HSP90 from normal cells.

3-Cyano-7-ethoxycoumarin
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3-Cyano-7-ethoxycoumarin

$105.00$245.00

3-Cyano-7-ethoxycoumarin is a fluorogenic cytochrome P-450 substrate that generates blue fluorescent product upon enzyme cleavage.

5-R-Rivaroxaban
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5-R-Rivaroxaban

$154.00$952.50

5-R-Rivaroxaban is (R) enantiomer of Rivaroxaban.

A 922500
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A 922500

$162.00$995.00

A 922500 is a potent, selective, and orally bioavailable DGAT-1 inhibitor with IC50 values of 7 nM and 24 nM for human and mouse DGAT-1 respectively.

A939572
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A939572

$525.00$840.00

A939572 (SCD1 inhibitor) is a potent, and orally bioavailable piperidine-aryl urea-based SCD1 inhibitor with IC50 values of <4 nM and 37 nM for mSCD1 and hSCD1 respectively.

Abiraterone
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Abiraterone

$182.00$351.00

Abiraterone (CB-7598) is a potent steroidal cytochrome P450 17alpha-hydroxylase-17,20-lyase (CYP17) inhibitor with an IC50 at 4 nM.

Abiraterone (acetate)
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Abiraterone (acetate)

$105.00$136.00

Abiraterone acetate (CB-7598) is a potent steroidal cytochrome P450 17alpha-hydroxylase-17,20-lyase (CYP17) inhibitor with an IC50 at 4 nM.

ABT-046
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ABT-046

$358.00$3,182.00

ABT-046 is a potent, selective, and orally bioavailable Diacylglycerol acyltransferase 1 (DGAT-1 ) inhibitor (IC50= 8 nM).

AEBSF
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AEBSF

$92.00$155.00

AEBSF is a water soluble, irreversible serine protease inhibitor; inhibits proteases like chymotrypsin, kallikrein, plasmin, thrombin, and trypsin.