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ARV-771 Chemical Structure Picture
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ARV-771

$246.00$3,386.00

ARV-771 is a potent bromodomain and extra-terminal (BET) proteins degrader based on PROTAC technology with Kd values of 4.7, 7.6, 7.6 nM against BRD2, BRD3 and BRD4, respectively.

ARV-825 Chemical Structure Picture
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ARV-825

$246.00$1,132.00

ARV-825 is a BRD4 Inhibitor based on PROTAC technology. ARV-825 shows affinity to BD1 and BD2 of BRD4 with Kds of 90 and 28 nM, respectively.

AT6 Chemical Structure Picture
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AT6

$743.00$2,151.00

AT6 is a PROTAC AT1 analogue, which is a highly selective bromodomain (Brd4) degrader.

BETd-260 Chemical Structure Picture
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BETd-260

$608.00$3,225.00

BETd-260 is a potent BET degrader based on PROTAC technology, with an IC50 of 30 pM against BRD4 protein in RS4;11 leukemia cell line.

BRD4 degrader AT1 Chemical Structure Picture
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BRD4 degrader AT1

$461.00$2,822.00

BRD4 degrader AT1 is a highly selective Brd4 degrader based on PROTAC technology, with a Kd of 44 nM for Brd4BD2 in cells.

dBET1 Chemical Structure Picture
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dBET1

$134.00$2,259.00

dBET1 is a potent BRD4 protein degrader based on PROTAC technology with an EC50 of 430 nM.

E3 ligase Ligand 1 Chemical Structure Picture
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E3 ligase Ligand 1

$407.00$2,420.00

E3 ligase Ligand 1 is a Ligand for E3 Ligase extracted from patent WO/2017/030814A1 compound example 202, used in PROTAC technology.

E3 ligase Ligand 1A Chemical Structure Picture
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E3 ligase Ligand 1A

$407.00$2,420.00

E3 ligase Ligand 1A is a ligand of E3 ligase, used in PROTAC technology; E3 ligase Ligand 1A can be used in the research of cancer.

E3 ligase Ligand 2 Chemical Structure Picture
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E3 ligase Ligand 2

$541.00$3,494.00

E3 ligase Ligand 2 is a Ligand for E3 Ligase used in PROTAC technology.

E3 ligase Ligand 3 Chemical Structure Picture
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E3 ligase Ligand 3

$541.00$3,494.00

E3 ligase Ligand 3 is a ligand of E3 ligase, used in PROTAC technology.

E3 ligase Ligand 4 Chemical Structure Picture
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E3 ligase Ligand 4

$541.00$3,494.00

E3 ligase Ligand 4 is a ligand of E3 ligase, used in PROTAC technology.

E3 ligase Ligand 5 Chemical Structure Picture
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E3 ligase Ligand 5

$1,615.00$4,701.00

E3 ligase Ligand 5 is a ligand of E3 ligase, extracted from patent US 20160058872A1, Paragraph 0515. E3 ligase Ligand 5 can be used in PROTAC technology.