Home Products Protein Biology Small Molecule Inhibitors Membrane Transporter/Ion Channel

Showing 1–12 of 644 results

Show sidebar
(-)-Borneol Chemical Structure Picture
Close

(-)-Borneol

$85.00$93.00

(-)-Borneol has a highly efficacious positive modulating action at GABA receptor with an EC50 of 237 μM.

(-)-MK 801 (Maleate) Chemical Structure Picture
Close

(-)-MK 801 (Maleate)

$85.00$303.00

(-)-MK 801 Maleate is the enantiomer of (+)-MK-801. (+)-MK 801 Maleate is a potent, selective and non-competitive NMDA receptor antagonist.

(-)-Securinine Chemical Structure Picture
Close

(-)-Securinine

$85.00$286.00

(-)-Securinine is plant-derived alkaloid and also a GABAA receptor antagonist.

(-)-Sparteine (sulfate pentahydrate) Chemical Structure Picture
Close

(-)-Sparteine (sulfate pentahydrate)

$72.00$79.00

(-)-Sparteine sulfate pentahydrate is a class 1a antiarrhythmic agent and a sodium channel blocker. It is an alkaloid, can chelate the bivalents calcium and magnesium.

(+)-Bicuculline Chemical Structure Picture
Close

(+)-Bicuculline

$102.00$310.00

(+)-Bicuculline, a convulsant alkaloid, is the antagonist of GABA.

(+)-Borneol Chemical Structure Picture
Close

(+)-Borneol

$117.00$128.00

(+)-Borneol (d-Borneol) is a natural bicyclic monoterpene used for analgesia and anesthesia in traditional Chinese medicine; enhances GABA receptor activity with an EC50 of 248 μM.

(+)-MK 801 (Maleate) Chemical Structure Picture
Close

(+)-MK 801 (Maleate)

$85.00$303.00

(+)-MK 801 (Maleate) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.

(+)-SJ733 Chemical Structure Picture
Close

(+)-SJ733

$310.00$6,767.00

(+)-SJ733 is a clinical candidate for malaria which can also inhibit Na+-ATPase PfATP4.

(+)-Tetrabenazine D6 Chemical Structure Picture
Close

(+)-Tetrabenazine D6

$380.00$1,615.00

(+)-Tetrabenazine D6 is the deuterium labeled (+)-Tetrabenazine. (+)-Tetrabenazine is a reversible inhibitor of vesicular monoamine transporter 2 (VMAT-2).

(20S)-Protopanaxadiol Chemical Structure Picture
Close

(20S)-Protopanaxadiol

$123.00$400.00

(20S)-Protopanaxadiol (20-Epiprotopanaxadiol) is an aglycon metabolic derivative of the protopanaxadiol-type ginseng saponin; apoptosis inducer.

(R)-Baclofen Chemical Structure Picture
Close

(R)-Baclofen

$85.00$295.00

(R)-Baclofen(STX209) is a selective GABAB receptor agonist. IC50 value:

(R)-Baclofen (hydrochloride) Chemical Structure Picture
Close

(R)-Baclofen (hydrochloride)

$85.00$295.00

(R)-Baclofen Hcl(STX-209 Hcl) is a derivative of gamma-aminobutyric acid (GABA) primarily used to treat spasticity and is in the early research stages for use for the treatment of alcoholism.