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(S)-(-)-5-Fluorowillardiine Chemical Structure Picture
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(S)-(-)-5-Fluorowillardiine

$239.00$954.00

(S)-(-)-5-Fluorowillardiine is a potent and specific AMPAR agonist.

7-Aminocephalosporanic acid Chemical Structure Picture
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7-Aminocephalosporanic acid

$102.00$111.00

7-Aminocephalosporanic acid is the core chemical structure for the synthesis of cephalosporin antibiotics, is a potent β-lactamase inhibitor.

7ACC1 Chemical Structure Picture
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7ACC1

$142.00$222.00

7ACC1(DEAC; Coumarin D 1421; D 1421) selectively interfere with lactate fluxes in the lactate-rich tumor microenvironment; inhibits lactate influx but not efflux in tumor cells expressing MCT1 and MCT4 transporters.

7ACC2 Chemical Structure Picture
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7ACC2

$263.00$3,386.00

7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for inhibition of [14C]-lactate influx; new antitumor treatment targeting lactate transport in cancer cells.

Acalisib Chemical Structure Picture
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Acalisib

$149.00$939.00

Acalisib is a potent and selective PI3Kδ inhibitor with an IC50 of 12.7 nM.

Acetaminophen Chemical Structure Picture
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Acetaminophen

$85.00$134.00

Acetaminophen (paracetamol) is a selective cyclooxygenase-2 (COX-2) inhibitor with an IC50 of 25.8 μM; is a widely used antipyretic and analgesic drug.

APD668 Chemical Structure Picture
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APD668

$246.00$2,259.00

APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119 respectively..

AR 231453 Chemical Structure Picture
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AR 231453

$120.00$180.00

AR231453 is a potent and selective small molecule agonist of GPR119 that enhances glucose-dependent insulin secretion and glucagon-like peptide 1 (GLP-1) release; Antidiabetic agent.

AT7519 Chemical Structure Picture
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AT7519

$85.00$341.00

AT7519 as a potent inhibitor of CDKs, with IC50s of 210, 47, 100, 13, 170, and <10 nM for CDK1, CDK2, CDK4 to CDK6, and CDK9, respectively.

AT7519 (Hydrochloride) Chemical Structure Picture
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AT7519 (Hydrochloride)

$85.00$341.00

AT7519 Hydrochloride is a potent inhibitor of CDKs, with IC50s of 210, 47, 100, 13, 170, and <10 nM for CDK1, CDK2, CDK4 to CDK6, and CDK9, respectively.

AT7519 (trifluoroacetate) Chemical Structure Picture
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AT7519 (trifluoroacetate)

$85.00$341.00

AT7519 trifluoroacetate as a potent inhibitor of CDKs, with IC50s of 210, 47, 100, 13, 170, and <10 nM for CDK1, CDK2, CDK4 to CDK6, and CDK9, respectively.

ATP-polyamine-biotin Chemical Structure Picture
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ATP-polyamine-biotin

$729.00$2,259.00

APB is a cell-permeable, efficient kinase cosubstrate with conversions and kinetics similar to those of other known ATP analogues. APB shows a cytotoxicity EC50 value of 19 ± 1 mM.